Product Name :
GR 103691
Description:
GR 103691 is a potent, selective dopamine D3 receptor antagonist with a Ki value of 0.4 nM. GR 103691 shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites.
CAS:
162408-66-4
Molecular Weight:
485.62
Formula:
C30H35N3O3
Chemical Name:
4′-acetyl-N-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl-[1,1′-biphenyl]-4-carboxamide
Smiles :
CC(=O)C1C=CC(=CC=1)C1C=CC(=CC=1)C(=O)NCCCCN1CCN(CC1)C1=CC=CC=C1OC
InChiKey:
JARNORYOPMINDY-UHFFFAOYSA-N
InChi :
InChI=1S/C30H35N3O3/c1-23(34)24-9-11-25(12-10-24)26-13-15-27(16-14-26)30(35)31-17-5-6-18-32-19-21-33(22-20-32)28-7-3-4-8-29(28)36-2/h3-4,7-16H,5-6,17-22H2,1-2H3,(H,31,35)
Purity:
≥98% (or refer to the Certificate of Analysis)
Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition :
Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.Galectin-4 Protein, Mouse (HEK293, His) Epigenetics
Shelf Life:
≥12 months if stored properly.
Stock Solution Storage:
0 – 4 oC for 1 month or refer to the Certificate of Analysis.
Additional information:
GR 103691 is a potent, selective dopamine D3 receptor antagonist with a Ki value of 0.4 nM. GR 103691 shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites.Clobenpropit web |Product information|CAS Number: 162408-66-4|Molecular Weight: 485.PMID:32310387 62|Formula: C30H35N3O3|Chemical Name: 4′-acetyl-N-4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl-[1,1′-biphenyl]-4-carboxamide|Smiles: CC(=O)C1C=CC(=CC=1)C1C=CC(=CC=1)C(=O)NCCCCN1CCN(CC1)C1=CC=CC=C1OC|InChiKey: JARNORYOPMINDY-UHFFFAOYSA-N|InChi: InChI=1S/C30H35N3O3/c1-23(34)24-9-11-25(12-10-24)26-13-15-27(16-14-26)30(35)31-17-5-6-18-32-19-21-33(22-20-32)28-7-3-4-8-29(28)36-2/h3-4,7-16H,5-6,17-22H2,1-2H3,(H,31,35)|Technical Data|Appearance: Solid Power|Purity: ≥98% (or refer to the Certificate of Analysis)|Solubility: DMSO : 25 mg/mL (51.48 mM; Need ultrasonic).|Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis|Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.|Shelf Life: ≥12 months if stored properly.|Stock Solution Storage: 0 – 4 oC for 1 month or refer to the Certificate of Analysis.|Drug Formulation: To be determined|HS Tariff Code: 382200|How to use|In Vitro:|GR 103691 shows marked affinity for serotonin1A (5-HT1A) receptors (Ki of 5.8 nM) and α-1 adrenoceptors (Ki of 12.6 nM).|Products are for research use only. Not for human use.|
